Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50162062(2-(5-Iodo-pyridin-3-yl)-7-methyl-7-aza-bicyclo[2.2...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha4-beta2 in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Brookhaven National Laboratory

Curated by ChEMBL
LigandPNGBDBM50177228(7-methyl-2-exo-(3'-iodo-5'-pyridinyl)-7-azabicyclo...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]epibatidine from alpha-4-beta-2 ACHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50162062(2-(5-Iodo-pyridin-3-yl)-7-methyl-7-aza-bicyclo[2.2...)
Affinity DataKi:  33nMAssay Description:Inhibition of [125I]-iodo-MLA binding to Nicotinic acetylcholine receptor alpha-7 in rat cerebral cortex More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed