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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Muscarinic acetylcholine receptor M3
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50223988
(8-methyl-8-aza-bicyclo[3.2.1]octan-3-yl benzyl(phe...)
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Affinity Data
IC50: 74.5nM
Assay Description:
Antagonist activity at cloned muscarinic M3 receptor expressed in CHO cells by measuring calcium mobilization
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50223988
(8-methyl-8-aza-bicyclo[3.2.1]octan-3-yl benzyl(phe...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 161nM
Assay Description:
Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells by measuring calcium mobilization
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50223988
(8-methyl-8-aza-bicyclo[3.2.1]octan-3-yl benzyl(phe...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 254nM
Assay Description:
Antagonist activity at cloned muscarinic M2 receptor expressed in CHO cells by measuring calcium mobilization
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI