Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM175375(1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-...)
BDBM175375(1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-...)
Ki: 3.99E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
BDBM175375(1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-...)
Ki: 6.38E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
BDBM175375(1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-...)
Ki: >3.00E+4nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair