Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
IC50: 68nMAssay Description:Inhibitory concentration for inhibition of Opioid receptor mu 1 induced contractions in guinea pig ileum (GPI) smooth muscle assaysMore data for this Ligand-Target Pair
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
BDBM50140910(19-methyl-(2R,10R)-11-oxa-8,19-diazahexacyclo[10.9...)
EC50: 3.00E+3nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudateMore data for this Ligand-Target Pair