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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of New Orleans

Curated by ChEMBL
LigandPNGBDBM50083533(4-(4-Chloro-phenyl)-1-methyl-piperidine-4-carbonit...)
Affinity DataKi:  5.11E+3nMAssay Description:Inhibition of [3H]paroxetine binding to rat serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of New Orleans

Curated by ChEMBL
LigandPNGBDBM50083533(4-(4-Chloro-phenyl)-1-methyl-piperidine-4-carbonit...)
Affinity DataKi:  5.11E+3nMAssay Description:Displacement of [3H]-paroxetine from serotonin transporter (SERT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of New Orleans

Curated by ChEMBL
LigandPNGBDBM50083533(4-(4-Chloro-phenyl)-1-methyl-piperidine-4-carbonit...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [3H]-WIN- 35,428 from dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of New Orleans

Curated by ChEMBL
LigandPNGBDBM50083533(4-(4-Chloro-phenyl)-1-methyl-piperidine-4-carbonit...)
Affinity DataKi:  2.20E+4nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New Orleans

Curated by ChEMBL
LigandPNGBDBM50083533(4-(4-Chloro-phenyl)-1-methyl-piperidine-4-carbonit...)
Affinity DataKi:  3.68E+4nMAssay Description:Inhibition of [3H]DAMGO binding to mu-opioid receptor at 100 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed