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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50089128(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-thiazol-2-yl...)
Affinity DataIC50:  450nMAssay Description:Inhibition of murine p38 alpha MAP kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50089128(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-thiazol-2-yl...)
Affinity DataIC50:  450nMAssay Description:Inhibition of murine phosphorylated His-Mitogen-activated protein kinase p38 alpha.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50089128(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-thiazol-2-yl...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1, COX-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed