Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMuscarinic acetylcholine receptor M2(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407329(CHEMBL2112938)
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 was determined by measuring its ability to displace [3H]-AF-DX 384 from rat he...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407329(CHEMBL2112938)
Affinity DataKi:  21.7nMAssay Description:In vitro binding affinity towards Sigma receptor type 1 was determined by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig brai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407329(CHEMBL2112938)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 was determined by measuring its ability to displace [3H]-Pirenzepine from bovi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407329(CHEMBL2112938)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- scopolamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed