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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

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TargetMuscarinic acetylcholine receptor M1(RAT)
Institute For Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50044689(2-(8-Methyl-2,4-dioxo-1-oxa-3,8-diaza-spiro[4.5]de...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]pirenzepine from rat cortex membrane expressing muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed