Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029793(8-[1-Cyclopropyl-meth-(E)-ylidene]-5-(3-hydroxy-ph...)
Affinity DataKi:  11.2nMAssay Description:Ability to inhibit [3H]-DAMGO binding to rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029793(8-[1-Cyclopropyl-meth-(E)-ylidene]-5-(3-hydroxy-ph...)
Affinity DataKi:  62.3nMAssay Description:Ability to inhibit [3H]-(+)-pentazocine binding to guinea pig brain Sigma receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029793(8-[1-Cyclopropyl-meth-(E)-ylidene]-5-(3-hydroxy-ph...)
Affinity DataKi: >500nMAssay Description:Ability to inhibit [3H]-U69,593 binding to guinea pig Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029793(8-[1-Cyclopropyl-meth-(E)-ylidene]-5-(3-hydroxy-ph...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to inhibit [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed