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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 16 hits in this display   

TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  9.40nMAssay Description:Ability to inhibit [3H]-(+)-pentazocine binding to guinea pig brain Sigma receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  9.40nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  9.40nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  9.40nMAssay Description:Ability to inhibit [3H]-(+)-pentazocine binding to guinea pig brain Sigma receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  23.3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  33.9nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  33.9nMAssay Description:Ability to inhibit [3H]-DAMGO binding to rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  392nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  392nMAssay Description:Ability to inhibit [3H]-DAMGO binding to rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi: >500nMAssay Description:Ability to inhibit [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi: >500nMAssay Description:Ability to inhibit [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi: >500nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  576nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  889nMAssay Description:Ability to inhibit [3H]-U69,593 binding to guinea pig Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  889nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  1.98E+3nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed