Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

LigandPNGBDBM50280553(8-Methyl-2,2-diphenyl-1,3-dioxa-8-aza-spiro[4.5]de...)
Affinity DataKi:  0.600nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280553(8-Methyl-2,2-diphenyl-1,3-dioxa-8-aza-spiro[4.5]de...)
Affinity DataKi:  8.10nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article