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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Muscarinic acetylcholine receptor M1
(RAT)
Universit£
Curated by
ChEMBL
Ligand
BDBM50062451
(3-(4-Methyl-piperazin-1-yl)-5-phenyl-pyridazine; h...)
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Affinity Data
Ki: 6.20E+4nM
Assay Description:
Compound was evaluated for its binding affinity for Muscarinic acetylcholine receptor M1 by measuring displacement of [3H]- pirenzepine from rat hipp...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Muscarinic acetylcholine receptor M2
(RAT)
Universit£
Curated by
ChEMBL
Ligand
BDBM50062451
(3-(4-Methyl-piperazin-1-yl)-5-phenyl-pyridazine; h...)
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Affinity Data
Ki: 8.00E+4nM
Assay Description:
Compound was evaluated for its binding affinity for Muscarinic acetylcholine receptor M2 by measuring displacement of [3H]- NMS ligand from rat cardi...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM50062451
(3-(4-Methyl-piperazin-1-yl)-5-phenyl-pyridazine; h...)
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Affinity Data
IC50: 36nM
Assay Description:
Compound was evaluated for its binding affinity for 5-hydroxytryptamine 3 receptor by measuring displacement of [3H]granisetron from rat cerebral cor...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI