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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50330508
(5-(4-Methylpiperazin-1-yl)-3-tosyl-1H-indazole | C...)
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Affinity Data
Ki: 4.90nM
Assay Description:
Displacement of [3H]LSD from human cloned 5HT6 receptor expressed in human HeLa cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50330508
(5-(4-Methylpiperazin-1-yl)-3-tosyl-1H-indazole | C...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 112nM
Assay Description:
Antagonist activity at human cloned 5HT6 receptor expressed in human HeLa cells by cyclase assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI