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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by
ChEMBL
Ligand
BDBM50304000
(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
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Affinity Data
Ki: 27nM
Assay Description:
Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of seratonin-induced cAMP accumulation by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by
ChEMBL
Ligand
BDBM50304000
(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
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Copy InChI
Affinity Data
Ki: 36.2nM
Assay Description:
Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by
ChEMBL
Ligand
BDBM50304000
(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >500nM
Assay Description:
Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI