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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
Astrazeneca R&D
Curated by
ChEMBL
Ligand
BDBM50179643
(1-(3-chlorophenyl)-3-(3-methylthiazolidin-2-yliden...)
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Affinity Data
IC50: 260nM
Assay Description:
Inhibition of glutamate-induced calcium influx in human mGluR5d by FLIPR
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Astrazeneca R&D
Curated by
ChEMBL
Ligand
BDBM50179643
(1-(3-chlorophenyl)-3-(3-methylthiazolidin-2-yliden...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.20E+3nM
Assay Description:
Displacement of [3H]MPEP from mGluR5d in rat brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI