Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 17 hits in this display
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
Ki: 7.90nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in rat cerebral cortical membrane using [3H]yohimbine as radioligand.More data for this Ligand-Target Pair
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
Ki: 100nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor in rat cerebral cortical membrane using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
BDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)