Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Vanderbilt Medical Center

Curated by ChEMBL

LigandBDBM50337959(2-((3-fluorophenyl)ethynyl)-6-methyl-7,8-dihydro-1...)Copy SMILESCopy InChI

Affinity DataIC50:  170nMAssay Description:Antagonist activity against mGlu5 receptor assessed as inhibition of calcium mobilizationMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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