Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
IC50: 20nMAssay Description:Inhibition of human PI3Kdelta (R108 to Q1044 residues) expressed in mammalian expression system incubated for 60 mins by ADAPTA assayMore data for this Ligand-Target Pair
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
IC50: 120nMAssay Description:Inhibition of human PI3Kgamma (S144 to A1102 residues) expressed in mammalian expression system incubated for 60 mins by ADAPTA assayMore data for this Ligand-Target Pair
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
IC50: 122nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
IC50: 355nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
BDBM50193016(CHEMBL3889977 | US11155556, No. 3)
IC50: 631nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair