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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNeutrophil collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286352((R)-2-(4-Benzyloxy-butyl)-N*1*-((S)-2,2-dimethyl-1...)
Affinity DataKi:  4.70nMAssay Description:Inhibition of human Matrix metalloproteinase-8More data for this Ligand-Target Pair
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TargetMatrix metalloproteinase-9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286352((R)-2-(4-Benzyloxy-butyl)-N*1*-((S)-2,2-dimethyl-1...)
Affinity DataKi:  11nMAssay Description:Inhibition of human Matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286352((R)-2-(4-Benzyloxy-butyl)-N*1*-((S)-2,2-dimethyl-1...)
Affinity DataKi:  39nMAssay Description:Inhibition of human fibroblast stromelysin, matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterstitial collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286352((R)-2-(4-Benzyloxy-butyl)-N*1*-((S)-2,2-dimethyl-1...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human fibroblast collagenase, matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails Article