Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215109((1R,3R,4R,7S)-(7-hydroxy-3-(adenin-9-yl)-2-oxa-5-a...)
Affinity DataIC50:  170nMAssay Description:Antagonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215109((1R,3R,4R,7S)-(7-hydroxy-3-(adenin-9-yl)-2-oxa-5-a...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed