Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246754(CHEMBL492599 | N'-{3-(R)-[2-(S)-(1H-Indol-3-yl)-1-...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human recombinant pro-MMP2 by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246754(CHEMBL492599 | N'-{3-(R)-[2-(S)-(1H-Indol-3-yl)-1-...)
Affinity DataIC50:  850nMAssay Description:Inhibition of human recombinant pro-MMP1 by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246754(CHEMBL492599 | N'-{3-(R)-[2-(S)-(1H-Indol-3-yl)-1-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant MMP14 catalytic domain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed