Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189015(1-(3-((S)-1-((R)-2-amino-3-(4-fluorophenyl)propano...)
Affinity DataKi:  261nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189015(1-(3-((S)-1-((R)-2-amino-3-(4-fluorophenyl)propano...)
Affinity DataKi:  461nMAssay Description:Binding affinity to human MC3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189015(1-(3-((S)-1-((R)-2-amino-3-(4-fluorophenyl)propano...)
Affinity DataKi:  2.13E+3nMAssay Description:Binding affinity to human MC1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189015(1-(3-((S)-1-((R)-2-amino-3-(4-fluorophenyl)propano...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed