Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040601((R)-2-[(S)-3-Methyl-1-((S)-1-methylcarbamoyl-2-phe...)
Affinity DataIC50:  49nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040601((R)-2-[(S)-3-Methyl-1-((S)-1-methylcarbamoyl-2-phe...)
Affinity DataIC50:  488nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040601((R)-2-[(S)-3-Methyl-1-((S)-1-methylcarbamoyl-2-phe...)
Affinity DataIC50:  2.34E+3nMAssay Description:Activity against human stromelysin (MMP-3).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed