Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50178305(ARCHAZOLID A)
Affinity DataKi:  967nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50178305(ARCHAZOLID A)
Affinity DataIC50:  86nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50178305(ARCHAZOLID A)
Affinity DataIC50:  352nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50178305(ARCHAZOLID A)
Affinity DataEC50:  200nMAssay Description:Agonist activity at farnesoid x receptor(unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed