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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetStromelysin-2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078171(CHEMBL3417770)
Affinity DataIC50:  12nMAssay Description:Inhibition of MMP-10 (unknown origin) measured every minute for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078171(CHEMBL3417770)
Affinity DataIC50:  15nMAssay Description:Inhibition of MMP-3 (unknown origin) measured every minute for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078172(CHEMBL3417769)
Affinity DataIC50:  17nMAssay Description:Inhibition of MMP-10 (unknown origin) measured every minute for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078172(CHEMBL3417769)
Affinity DataIC50:  18nMAssay Description:Inhibition of MMP-3 (unknown origin) measured every minute for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078190(CHEMBL3417751)
Affinity DataIC50:  21nMAssay Description:Inhibition of MMP-10 (unknown origin) measured every minute for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078190(CHEMBL3417751)
Affinity DataIC50:  21nMAssay Description:Inhibition of MMP-3 (unknown origin) measured every minute for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078172(CHEMBL3417769)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG channel by patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078171(CHEMBL3417770)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG channel by patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078172(CHEMBL3417769)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG channel after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078190(CHEMBL3417751)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG channel after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Navarra

Curated by ChEMBL
LigandPNGBDBM50078171(CHEMBL3417770)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG channel after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed