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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50442973(CHEMBL3086285)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50442973(CHEMBL3086285)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed