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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Neurocrine Biosciences
Curated by
ChEMBL
Ligand
BDBM50150831
(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
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Affinity Data
Ki: 36nM
Assay Description:
Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Melanocortin receptor 4
(Homo sapiens (Human))
Neurocrine Biosciences
Curated by
ChEMBL
Ligand
BDBM50150831
(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.40E+3nM
Assay Description:
Binding affinity for human melanocortin 4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Neurocrine Biosciences
Curated by
ChEMBL
Ligand
BDBM50150831
(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.30E+3nM
Assay Description:
Binding affinity for human melanocortin 3 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Neurocrine Biosciences
Curated by
ChEMBL
Ligand
BDBM50150831
(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 630nM
Assay Description:
Inhibition of human Melanocortin 5 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Neurocrine Biosciences
Curated by
ChEMBL
Ligand
BDBM50150831
(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 4.60E+3nM
Assay Description:
Agonistic activity for human Melanocortin 4 receptor as stimulated cAMP release
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI