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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetProtein artemis(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM51800(4-(1H-indol-3-yl)-N-methyl-1,3-thiazol-2-amine | 4...)
Affinity DataIC50:  2.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM51800(4-(1H-indol-3-yl)-N-methyl-1,3-thiazol-2-amine | 4...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM51800(4-(1H-indol-3-yl)-N-methyl-1,3-thiazol-2-amine | 4...)
Affinity DataEC50:  4.99E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM51800(4-(1H-indol-3-yl)-N-methyl-1,3-thiazol-2-amine | 4...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetXylosyl- and glucuronyltransferase LARGE1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM51800(4-(1H-indol-3-yl)-N-methyl-1,3-thiazol-2-amine | 4...)
Affinity DataEC50:  1.03E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay