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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Tyrosine-protein kinase Mer
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50384597
(CHEMBL2036633 | US9744172, Compound UNC00000486A)
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Affinity Data
IC50: 170nM
Assay Description:
Inhibition of Mer expressed in Escherichia coli BL21 (DE3) cells using EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluid capillary electr...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50384597
(CHEMBL2036633 | US9744172, Compound UNC00000486A)
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Copy InChI
Affinity Data
IC50: 220nM
Assay Description:
Inhibition of Axl using KKKKEEIYFFF-CONH2 as substrate after 180 mins by microfluid capillary electrophoresis assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase Mer
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50384597
(CHEMBL2036633 | US9744172, Compound UNC00000486A)
Copy SMILES
Copy InChI
Affinity Data
IC50: 550nM
Assay Description:
The ectopic expression of Mer receptor tyrosine kinase (Mer) has been identified as a tumor cell survival gene product in Acute Lymphoblastic Leukemi...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Tyrosine-protein kinase receptor TYRO3
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50384597
(CHEMBL2036633 | US9744172, Compound UNC00000486A)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.10E+3nM
Assay Description:
Inhibition of Tyro3 using EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluid capillary electrophoresis assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI