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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Chemical Diversity Research Institute
Curated by
ChEMBL
Ligand
BDBM50318627
(CHEMBL1083075 | N,5-Dimethyl-3-(phenylsulfonyl)-7,...)
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Affinity Data
Ki: 0.202nM
Assay Description:
Displacement of [3H]lysergic acid diethylamide from human recombinant 5HT6 receptor expressed in human HeLa cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
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Ligand Info
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Chemical Diversity Research Institute
Curated by
ChEMBL
Ligand
BDBM50318627
(CHEMBL1083075 | N,5-Dimethyl-3-(phenylsulfonyl)-7,...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.413nM
Assay Description:
Antagonist activity at human 5HT6 receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced cAMP release
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Chemical Diversity Research Institute
Curated by
ChEMBL
Ligand
BDBM50318627
(CHEMBL1083075 | N,5-Dimethyl-3-(phenylsulfonyl)-7,...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 188nM
Assay Description:
Antagonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as inhibition of alpha-Me-serotonin-induced intracellular calcium mobi...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI