Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Apelin receptor
(Homo sapiens (Human))
Amgen
US Patent
Ligand
BDBM269998
((1R,2S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.30nM
pH: 7.5
Assay Description:
The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Apelin receptor
(Homo sapiens (Human))
Amgen
US Patent
Ligand
BDBM269998
((1R,2S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.30nM
Assay Description:
The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Apelin receptor
(Homo sapiens (Human))
Amgen
US Patent
Ligand
BDBM269998
((1R,2S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.30nM
Assay Description:
The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI