Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetStromelysin-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131664(CHEMBL326489 | N*4*-Hydroxy-N*1*-{1-[(methoxy-phen...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131664(CHEMBL326489 | N*4*-Hydroxy-N*1*-{1-[(methoxy-phen...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131664(CHEMBL326489 | N*4*-Hydroxy-N*1*-{1-[(methoxy-phen...)
Affinity DataIC50:  750nMAssay Description:Inhibition of human matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131664(CHEMBL326489 | N*4*-Hydroxy-N*1*-{1-[(methoxy-phen...)
Affinity DataIC50:  930nMAssay Description:Inhibition of Matrix metalloprotease-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50131664(CHEMBL326489 | N*4*-Hydroxy-N*1*-{1-[(methoxy-phen...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed