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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50321777((R)-1'-benzyl-6-methoxy-1-phenyl-1,6-dihydrospiro[...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50321777((R)-1'-benzyl-6-methoxy-1-phenyl-1,6-dihydrospiro[...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50321777((R)-1'-benzyl-6-methoxy-1-phenyl-1,6-dihydrospiro[...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50321777((R)-1'-benzyl-6-methoxy-1-phenyl-1,6-dihydrospiro[...)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50321777((R)-1'-benzyl-6-methoxy-1-phenyl-1,6-dihydrospiro[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of 5HTT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50321777((R)-1'-benzyl-6-methoxy-1-phenyl-1,6-dihydrospiro[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed