Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
EC50: 41nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
EC50: 2.70nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
EC50: 0.280nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
EC50: 41nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
EC50: 2.70nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM270006((1S,2R)-1-(5-cyano-2-pyridinyl)-N-(4-(2,6-dimethox...)
EC50: 41nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair