Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116720(CHEMBL77042 | [3-(1-{(R)-5-[(3,5-Dichloro-benzoyl)...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against recombinant human tachykinin receptor 1 in CHO cells using [3H]-Sar SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116720(CHEMBL77042 | [3-(1-{(R)-5-[(3,5-Dichloro-benzoyl)...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity against recombinant human tachykinin receptor 2 in CHO cells using [3H]-NKA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116720(CHEMBL77042 | [3-(1-{(R)-5-[(3,5-Dichloro-benzoyl)...)
Affinity DataKi:  11nMAssay Description:Binding affinity against recombinant human tachykinin receptor 3 in CHO cells using [125I]-[MePhe]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed