Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 22 hits in this display
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
IC50: 45nMAssay Description:The MLK1, MLK2, and MLK3 assays were performed using the Millipore multiscreen trichloroacetic acid (TCA) in-plate format. IC50 values were calculate...More data for this Ligand-Target Pair
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
IC50: 150nMpH: 7.6 T: 2°CAssay Description:A coupled-enzyme assay was used to quantify the ADP generated in the kinase reaction with S6 peptide (RRRLSSLRA) as the phosphoacceptorsubstrate.More data for this Ligand-Target Pair
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
BDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)