Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50334059((2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-((S)-2-amino...)
Affinity DataKi:  3.78E+3nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50166732((3S,4aR,6S,8R,8aR)-6-((S)-2-Amino-propionyloxy)-3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor kappa 1 expressed in chinese hamster ovary cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50334059((2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-((S)-2-amino...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50334059((2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-((S)-2-amino...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed