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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Aminopeptidase N
(Sus scrofa (Pig))
Shandong University
Ligand
BDBM235702
(L-Isoseryl-L-leucyl-L-phenylalanine benzyl ester h...)
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Affinity Data
IC50: 6.91E+4nM
Assay Description:
The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
72 kDa type IV collagenase
(Homo sapiens (Human))
Shandong University
Ligand
BDBM235702
(L-Isoseryl-L-leucyl-L-phenylalanine benzyl ester h...)
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Affinity Data
IC50: 2.37E+5nM
pH: 8.5 T: 2°C
Assay Description:
The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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