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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Bromodomain testis-specific protein [21-137]
(Homo sapiens (Human))
Dana-Farber Cancer Institute
Ligand
BDBM205434
((6S+2S)-PEG4 (10))
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Affinity Data
IC50: 1.09nM
pH: 7.5 T: 2°C
Assay Description:
Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Bromodomain-containing protein 4 [44-168]
(Homo sapiens (Human))
Dana-Farber Cancer Institute
Ligand
BDBM205434
((6S+2S)-PEG4 (10))
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Copy InChI
Affinity Data
IC50: 2.95nM
pH: 7.5 T: 2°C
Assay Description:
Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168]
(Homo sapiens (Human))
Dana-Farber Cancer Institute
Ligand
BDBM205434
((6S+2S)-PEG4 (10))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.0230nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4 [44-168,333-460]
(Homo sapiens (Human))
Dana-Farber Cancer Institute
Ligand
BDBM205434
((6S+2S)-PEG4 (10))
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.00660nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI