Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 86 hits in this display
BDBM50005539((3S,8R)-8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50005539((3S,8R)-8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50156919((2R,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50005539((3S,8R)-8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50156919((2R,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50156923((1R)-3-alpha-(4-methylphenyl)tropane-2-alpha-carbo...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50156919((2R,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50156923((1R)-3-alpha-(4-methylphenyl)tropane-2-alpha-carbo...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
IC50: 26nMAssay Description:Inhibitory activity against Serotonin transporter was determined for [3H]5-HT (serotonin) uptake by striated synaptosomesMore data for this Ligand-Target Pair
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50039990((3S,8R)-8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50156919((2R,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50156923((1R)-3-alpha-(4-methylphenyl)tropane-2-alpha-carbo...)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50006781((2S,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50156923((1R)-3-alpha-(4-methylphenyl)tropane-2-alpha-carbo...)
BDBM50156919((2R,3S)-methyl 8-methyl-3-p-tolyl-8-aza-bicyclo[3....)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
BDBM50035729(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane | 8-...)
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