Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
Ki: 50nMAssay Description:Inhibition of human recombinant MMP-2 using MOCAcPLGLA2pr(Dnp)AR-NH2 as substrate by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
Ki: 180nMAssay Description:Inhibition of human recombinant MMP-9 catalytic domain using MOCAcPLGLA2pr(Dnp)AR-NH2 as substrate by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
Ki: 2.60E+3nMAssay Description:Inhibition of human recombinant MMP-14 catalytic domain using MOCAcPLGLA2pr(Dnp)AR-NH2 as substrate by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
Ki: 1.30E+4nMAssay Description:The term selective inhibitor as used in reference to MMPs refers to an inhibitor that inhibits the enzymatic activity of one MMP in the presence of o...More data for this Ligand-Target Pair
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
Ki: 1.30E+4nMAssay Description:Inhibition of human recombinant MMP-8 catalytic domain using McaKPLGL9(Dpa)AR-NH2 as substrate by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
BDBM50442356(CHEMBL2442885 | US10357546, ND-380 | US9951035, ND...)
Ki: 1.30E+4nMAssay Description:Human recombinant active MMP-2 and MMP-7, and the catalytic domains of MMP-3 and MMP-14/MT1-MMP were purchased from EMD Chemicals, Inc. (San Diego, C...More data for this Ligand-Target Pair