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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
Sanford-Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM46005(4-methoxy-3-(3-quinolinylsulfamoyl)benzoic acid me...)
Affinity DataIC50:  550nMAssay Description:To determine the inhibition selectivity for inhibitor candidates, human TNAP, PLAP or IAP were added to microtiter plates followed by addition of the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Homo sapiens (Human))
Sanford-Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM46005(4-methoxy-3-(3-quinolinylsulfamoyl)benzoic acid me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay