Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50316703(CHEMBL1094545 | N-[2-(7-{4-[4'-Methoxycarbonylbiph...)
Affinity DataKi:  2.40nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50316703(CHEMBL1094545 | N-[2-(7-{4-[4'-Methoxycarbonylbiph...)
Affinity DataKi:  19nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50316703(CHEMBL1094545 | N-[2-(7-{4-[4'-Methoxycarbonylbiph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human human MT2 receptor expressed in CHO cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50316703(CHEMBL1094545 | N-[2-(7-{4-[4'-Methoxycarbonylbiph...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human human MT1 receptor expressed in CHO cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed