Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50182459(CHEMBL201717 | methyl 4'-[({2-methyl-2-[(3,3,3-tri...)
Affinity DataKi:  3.45E+3nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50182459(CHEMBL201717 | methyl 4'-[({2-methyl-2-[(3,3,3-tri...)
Affinity DataKi:  3.50E+3nMAssay Description:Antagonist activity at Bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50182459(CHEMBL201717 | methyl 4'-[({2-methyl-2-[(3,3,3-tri...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to bradykinin B2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed