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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM98036(US8486953, 19)
Affinity DataKi:  4.05E+3nMAssay Description:Inhibition of human Mnk2a using TAMRA-labeled eIF4E peptide as substrate incubated for 10 mins followed by addition of ATP measured after 90 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM98036(US8486953, 19)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk1a (unknown origin) using TAMRA-labeled eIF4E peptide as substrate incubated for 10 mins followed by addition of ATP measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM98036(US8486953, 19)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of CDK2/cyclinA (unknown origin) using TAMRA-labeled eIF4E peptide as substrate incubated for 10 mins followed by addition of ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM98036(US8486953, 19)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of CDK9/cyclinT1 (unknown origin) using TAMRA-labeled eIF4E peptide as substrate incubated for 10 mins followed by addition of ATP measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM98036(US8486953, 19)
Affinity DataIC50:  4nMpH: 7.4 T: 2°CAssay Description:Inhibition of kinase activity of Mnk1 and Mnk2a was assessed with the same assay system, using pre-activated GST-Mnk1 or GST-Mnk2a, respectively. The...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM98036(US8486953, 19)
Affinity DataIC50:  60nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM98036(US8486953, 19)
Affinity DataIC50:  590nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent