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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50091723
((S)-3-{(1R,3S)-3-[4-(2-Cyano-phenyl)-piperidin-1-y...)
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Affinity Data
Ki: 0.240nM
Assay Description:
Displacement of [125I]HEAT from human Alpha-1A adrenergic receptor stably expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50091723
((S)-3-{(1R,3S)-3-[4-(2-Cyano-phenyl)-piperidin-1-y...)
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Copy InChI
Affinity Data
Ki: 16nM
Assay Description:
Displacement of [125I]HEAT from human Alpha-1D adrenergic receptor stably expressed in HL cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50091723
((S)-3-{(1R,3S)-3-[4-(2-Cyano-phenyl)-piperidin-1-y...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 130nM
Assay Description:
Displacement of [125I]HEAT from human Alpha-1B adrenergic receptor stably expressed in LM cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI