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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
11
hits in this display
Target
Prothrombin
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 0.00700nM
Assay Description:
Binding affinity against alpha thrombin
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Prothrombin
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 0.0280nM
Assay Description:
Binding affinity against gamma thrombin
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Serine protease 1
(Bos taurus (bovine))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 0.670nM
Assay Description:
Binding affinity against Trypsin
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Chymotrypsinogen A
(Bos taurus (bovine))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 1.21nM
Assay Description:
Binding affinity against Chymotrypsin
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Chymotrypsin-like elastase family member 2A
(Sus scrofa)
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 3.08nM
Assay Description:
Binding affinity of the compound towards porcine pancreatic elastase
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Coagulation factor X
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 3.10nM
Assay Description:
Binding affinity against Coagulation factor X
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Cathepsin G
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 3.90nM
Assay Description:
Binding affinity against cathepsin G
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Kallikrein-1
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 6.10nM
Assay Description:
Binding affinity against kallikrein
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Plasminogen
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 7.80nM
Assay Description:
Binding affinity against plasmin
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Urokinase-type plasminogen activator
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
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Affinity Data
Ki: 81nM
Assay Description:
Binding affinity against Urokinase plasminogen activator
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prothrombin
(Homo sapiens (Human))
Thrombosis Research Institute
Curated by
ChEMBL
Ligand
BDBM50034574
(CHEMBL288150 | Peptide boronate)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.10E+4nM
Assay Description:
Binding affinity against thrombin
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI