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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50106086((S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-prop...)
Affinity DataIC50:  7.10nMAssay Description:In vitro Very late antigen 4 cell adhesion inhibitory activity measured by binding of fluorescently labeled Ramos cells to immobilized VCAM-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50106086((S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-prop...)
Affinity DataIC50:  13nMAssay Description:Inhibition of fluorescent Ramos cell adhesion to fibronectin by Very late antigen 5 (VLA-5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50106086((S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-prop...)
Affinity DataIC50:  22nMAssay Description:Inhibition of fluorescent Ramos cell adhesion to VCAM-1 by rat Very late antigen 4 (VLA-4) integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50106086((S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-prop...)
Affinity DataIC50:  27nMAssay Description:Inhibition of fluorescent Ramos cell adhesion to VCAM-1 by mouse Very late antigen 4 (VLA-4) integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50106086((S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-prop...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of fluorescent Ramos cell adhesion to VCAM-1 by alpha4-beta7 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50106086((S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-prop...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of fluorescent Ramos cell adhesion to fibronectin by Very late antigen 4 (VLA-4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed