Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

LigandBDBM75184((E)-2-cyano-3-[4-keto-2-[4-(4-methoxyphenyl)pipera...)Copy SMILESCopy InChI

Affinity DataEC50: >6.95E+4nMMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In DepthDetails PCBioAssay
Copy BDB DOI

TargetImportin subunit alpha-1(Homo sapiens (Human))
Broad Institute

Curated by PubChem BioAssay

LigandBDBM75184((E)-2-cyano-3-[4-keto-2-[4-(4-methoxyphenyl)pipera...)Copy SMILESCopy InChI

Affinity DataEC50:  4.65E+4nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In DepthDetails PCBioAssay
Copy BDB DOI