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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  17nMAssay Description:Inhibition of p56lck autophosphorylationChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  17nMAssay Description:Inhibition of p56 Lck tyrosine kinase in Jurkat cells where p56lck autophosphorylation is inhibited.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  620nMAssay Description:Inhibition of p56lck-mediated exogenous peptide phosphorylationChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  800nMMore data for this Ligand-Target Pair
In DepthDetails
TargetLIM domain kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  800nMAssay Description:Inhibition of his6 tagged LIMK1 (unknown origin) expressed in baculovirus-infected Sf9 cells measured after 1 hr in presence of ATP by fluorescence b...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLIM domain kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  800nMAssay Description:Inhibition of Limk1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetLIM domain kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50366492(DAMNACANTHAL)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of his6 tagged LIMK2 (unknown origin) expressed in baculovirus-infected Sf9 cells measured after 1 hr in presence of ATP by fluorescence b...More data for this Ligand-Target Pair
In DepthDetails PubMed